Advanced SearchSearch Tips
Synthesis and Biological Evaluation of 2-Amino-4H-pyran-3,4,5-tricarboxylate Salt Derivatives
facebook(new window)  Pirnt(new window) E-mail(new window) Excel Download
 Title & Authors
Synthesis and Biological Evaluation of 2-Amino-4H-pyran-3,4,5-tricarboxylate Salt Derivatives
Akbari, Ali; Azami-Sardooei, Zabihollah; Hosseini-Nia, Asghar;
  PDF(new window)
A novel and simple method for the synthesis of 2-amino-4H-pyran-3,4,5-tricarboxylate derivative and the evaluation of their antibacterial activity against Pseudomonas syringae, Xanthomonas citi and Pectobacterium carotovorum are reported. The structure of the isolated compounds has been determined by means of NMR and FT-IR Spectroscopy. The reaction of alkyl isocyanides with acetylenic esters in the presence of dimethyl acetone-1,3-dicarboxylate in the present of at ambient temperature. Some of the compound showed significant inhibition to growth of bacteria.
Biological evaluation;Antibacterial activity;4H-Pyran-3;4;5-tricarboxylate;;
 Cited by
Synthesis of mesoporous Ca-MCM catalysts and their use in suitable multicomponent synthesis of polyfunctionalized pyrans, Research on Chemical Intermediates, 2017, 43, 4, 2103  crossref(new windwow)
Wilson, K.; Clark, J. H. Synthesis of a Novel Supported Solid Acid $BF_{3}$ Catalyst. Chem. Commun. 1998, 2135.

Klapotke, T. M.; Mc Monagle, F.; Spence, R. R.; Winfield, J. M. $\gamma$-Alumina-Supported Boron Trifluoride: Catalysis, Radiotracer Studies and Computations. J. Fluorine. Chem. 2006, 127, 1446. crossref(new window)

Sadegi, B.; Mirjalili, B. F.; Hashemi, M. M. $BF_{3}{\cdot}SiO_{2}$: An Efficient Reagent System for the One-Pot Synthesis of 1,2,4,5-Tetrasubstituted Imidazoles. Tetrahedron Lett. 2008, 49, 2575. crossref(new window)

Mirjalili, B. F.; Bamoniri, A.; Akbari, A. $BF_{3}{\cdot}SiO_{2}$: An Efficient Alternative for the Synthesis of 14-Aryl or Alkyl-14H-dibenzo[a,j]xanthenes. Tetrahedron Lett. 2008, 49, 6454. crossref(new window)

Sadegi, B.; Mirjalili, B. F.; Hashememi, M. M. $BF_{3}{\cdot}SiO_{2}$: An Efficient Heterogeneous Alternative for Regio-Chemo and Stereoselective Claisen-schmidt Condensation. J. Iran. Chem. Soc. 2008, 5(4), 694. crossref(new window)

Boodhoo, K. V. K.; Dunk, W. A. E.; Vicevic, M.; Jachuck, R. J.; Sage, V.; Macquarrie, D. J.; Clark, J. H. Classical Cationic Polymerisation of Styrene in a Spinning Disc Reactor Using Silica Supported $BF_{3$ Catalyst. J. Appl. Polym. Sci. 2006, 101(1), 8. crossref(new window)

Dindulkar, S. D.; Parthiban P.; Y. T. Jeong. $BF_{3}{\cdot}SiO_{2}$ is a Simple and Efficient Lewis Acid Catalyst for the One-Pot Synthesis of Polyfunctionalized Piperidin-4-ones. Monatsh. Chem. 2012, 143, 113. crossref(new window)

Reddy, M. V.; Dindulkar, S. D.; Jeong, Y. T. $BF_{3}{\cdot}SiO_{2}$- Catalyzed One-Pot Synthesis of $\alpha$-Aminophosphonates in Ionic Liquid and Neat Conditions. Tetrahedron Lett. 2011, 52, 4764. crossref(new window)

Mirjalili, B. F.; Bamoniri, A.; Akbari, A. Nano-$BF_{3}{\cdot}SiO_{2}$: a Reusable and Eco-friendly Catalyst for Synthesis of Quinoxalines. Chem. Heterocycl. Comp. 2011, 47(4), 487. crossref(new window)

Mirjalili, B. F.; Bamoniri, A.; Akbari, A. One-pot Synthesis of 3,4-Dihydropyrimidin-2(1H)-ones (thiones) Promoted by Nano-$BF_{3}{\cdot}SiO_{2}$. J. Iran. Chem. Soc. 2011, 8, 135. crossref(new window)

Rho, H. S.; Baek, H. S.; You, J. W.; Kim, S.; Lee, J. Y.; Kim, D. H.; Chang, I. S. Bull. Korean Chem. Soc. 2007, 28(3), 471. crossref(new window)

Li, D.-H.; Cai, S.-X.; Tian, L.; Lin, Z.-J.; Zhu, T.-J.; Fang, Y.-C.; Liu, P.-P.; Gu, Q.-Q.; Zhu, W.-M. Arch. Pharm. Res. 2007, 30(9), 1051. crossref(new window)

Wang, T.-S.; Wang, S.-Q.; Xiao, D.-L. J. Med. Plants Res. 2012, 6(26), 4259.

Larget, R.; Lockhart, B.; Renard, P.; Largeron, M. Biorg. Med. Chem. Lett. 2000, 10, 835. crossref(new window)

Groweiss, A.; Cardellins, J. H.; Boyd, M. R. J. Nat. Prod. 2000, 63, 1537. crossref(new window)

Deng, Y.; Lee, J. P.; Ramamonjy, M. T.; Synder, J. K.; Des Etages, S. A.; Kanada, D.; Synder, M. P.; Turner, C. J. J. Nat. Prod. 2000, 63, 1082. crossref(new window)

Khan, I. A.; Avery, M. A.; Burandt, C. L.; Goins, D. K.; Mikell, J. R.; Nash, T. E.; Azadega, A.; Walker, L. A. J. Nat. Prod. 2000, 63, 1414. crossref(new window)

Mori, K.; Audran, G.; Monti, H. Synlett 1998, 259.

Pietta, P. J. J. Nat. Prod. 2000, 63, 1035. crossref(new window)

Nasiri, F.; Nazem, F.; Pourdavaie, K. Mol. Divers. 2007, 11, 101. crossref(new window)

Park, E.-J.; Gray, P. M.; Oh, S.-W.; Kronenberg, J.; Kang, D.-H. J. Food. Science. 2008, 73(6), M278. crossref(new window)

Toth, I. K.; Bell, K. S.; Holeva, M. C., Birch, P. R. J. Molecular Plant Pathology 2003, 4(1), 17. crossref(new window)

Yang, J. W.; Yi, H.-S.; Kim, H.; Lee, B.; Lee, S.; Ghim, S.-Y.; Ryu, C.-M. J. Ecology. 2011, 99(1), 46. crossref(new window)

Boch, J.; Bonas, U. Annual Review of Phytopathology 2010, 48, 419. crossref(new window)

Ivanovic, Z.; Zivkovic, S.; Starovic, M.; Josic, D.; Stankovic, S.; Gavrilovic, V. Arch. Biol. Sci. 2009, 61(4), 863. crossref(new window)

Rodrigo, J. Sci. Hortic. 2000, 85(3), 155. crossref(new window)

Lemriss, S.; Marquet, B.; Ginestet, H.; Lefeuvre, L.; Fassouane, A.; Boiron, P. J. Mycol. Med. 2003, 13, 189.

Rahman, A.; Choudhary, M. I.; Thomsen, W. J. Bioassay Techniques for Drug Development; Harwood Academic Publishers: Amsterdam, 2001; p 14.