Synthesis and fungicidal activity of new ${\beta}$-methoxyacrylate derivatives having thio-enol side chain

티오엔을 곁가지를 가진 메톡시아크릴레이트 화합물의 합성 및 살균활성 연구

  • Lee, Hyeon-Kyu (Bio-Organic Science Division, Korea Research Institute of Chemical Technology) ;
  • Kim, Ji-A (Bio-Organic Science Division, Korea Research Institute of Chemical Technology) ;
  • Choi, Eun-Bok (Bio-Organic Science Division, Korea Research Institute of Chemical Technology) ;
  • Park, Chwang-Siek (Bio-Organic Science Division, Korea Research Institute of Chemical Technology) ;
  • Choi, Gyung-Ja (Bio-Organic Science Division, Korea Research Institute of Chemical Technology)
  • 이현규 (한국화학연구원 생물화학연구부) ;
  • 김지아 (한국화학연구원 생물화학연구부) ;
  • 최은복 (한국화학연구원 생물화학연구부) ;
  • 박창식 (한국화학연구원 생물화학연구부) ;
  • 최경자 (한국화학연구원 생물화학연구부)
  • Published : 2005.06.30

Abstract

New ${\beta}$-methoxyacrylate derivatives 1-4 having thio-enol side chain were prepared and subjected to in vivo screening for fungicidal activity against phytopathogenic fungi and many of them showed good fungicidal activities against especially rice blast and wheat leaf rust at 100 ppm.

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