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Synthesis of Nucleophilic Adducts of Thiols (XI). Addition of L-Cysteine to $\beta,\beta$-Dinitrostyrene Derivatives

  • Kim, Tae-Rin (Department of Chemistry, Korea University) ;
  • Kim, Jae-Hoon (Department of Chemistry, Kum-Oh Institute of Technology) ;
  • Choi, Won-Sik (Department of Chemistry, Kangreung National University)
  • 발행 : 1988.06.20

초록

The addition of L-cysteine without blocking amino and carboxyl groups to${\beta},{\beta}$-dinitrostyrene derivatives(11a-e) were investigated. ${\beta},{\beta}$ -Dinitrostyrene derivatives(11a-e) easily undergo addition reactions with L-cysteine to from s-(2,2-dinitro-1-phenylethyl)-L-cysteine(12a), s-[2,2-dinitro-1-(p-methyl)phenylethyl]-L-cysteine (12b), s-[2,2-dinitro-1-(p-methoxy)phenylethyl]-L-cystein e(12c), s-[2,2-dinitro-1-(p-chloro)phenylethyl]-L-cysteine (12d) and s-[2,2-dinitro-1-(p-nitro)phenylethyl]-L-cysteine( 12a), respectively. The structure of adducts were confirmed by means of spectral data, molecular weight measurement and elemental analysis.

키워드

참고문헌

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피인용 문헌

  1. β,β-Dinitrostyrenes Reacted with Pyrrole vol.41, pp.5, 2005, https://doi.org/10.1007/s10593-005-0202-8
  2. Specific features of the reaction of β,β-dinitrostyrenes with indan-1,3-dione vol.76, pp.8, 1988, https://doi.org/10.1134/s1070363206080391
  3. β,β-Dinitrostyrenes in reactions with cyclohexane-1,3-diones vol.58, pp.10, 1988, https://doi.org/10.1007/s11172-009-0278-x