The Korean Journal of Pesticide Science (농약과학회지)

The Korean Society of Pesticide Science (한국농약과학회)
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Synthesis and herbicidal activities of 9-(5-isoxazolemethoxy-phenyl)imino-8-thia-1,6-diazabicyclo[4.3.0]nonan-7-one and their related derivatives

새로운 9-(5-isoxazolemethoxyphenyl)imino-8-thia-1,6-diazabicycio [4.3.0]nonan-7-one 유도체의 합성과 제초활성

  • Published : 2003.12.30
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Abstract

New series of 9-(5-Isoxazolemethoxyphenyl)imino-8-thia-l,6-diazabicyclo[4.3.0]nonan-7-one which are the cyclic imide type compounds were designed and synthesized. The herbicidal activities of main dominant weeds to these compounds were evaluated under rice field condition. There is the possibility for a new herbicide since the most of compounds were excellent to main dominant weeds occurring in rice field without the serious rice injury.

고리형 이미드계 화합물 중에서 제초활성이 매우 좋을 것으로 예상된 9-(5-isoxazolemethoxypheny1) imino-8-thia-1,6-diazabicyclo[4.3.0]nonan-7-one 유도체들을 합성하였고 이들의 제초활성을 논조건에서 시험하였다. 대부분의 화합물의 제초활성은 매우 강하였으며 벼에는 약해가 거의 나타나지 않았다. 올챙이고랭이와 올미에 대해서는 활성이 약하였으나 피와 물달개비, 너도방동사니에 대해서 매우 좋은 제초활성을 보여 신규제초제로서 가능성을 보였다.

Keywords

References

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